BP501T MEDICINAL CHEMISTRY – II (Theory) Notes

5.1 Antidiabetic agents Insulin and its preparations Sulfonyl ureas: Tolbutamide*, Chlorpropamide, Glipizide, Glimepiride. Biguanides: Metformin. Thiazolidinediones: Pioglitazone, Rosiglitazone. Meglitinides: Repaglinide, Nateglinide. Glucosidase inhibitors: Acrabose, Voglibose. Please follow the link  Antidiabetic agents

Local Anesthetics: SAR of Local anesthetics Benzoic Acid derivatives ; Cocaine, Hexylcaine, Meprylcaine, Cyclomethycaine,Piperocaine. Amino Benzoic acid derivatives : Benzocaine*, Butamben, Procaine*, Butacaine,Propoxycaine, Tetracaine, Benoxinate. Lidocaine/Anilide derivatives : Lignocaine, Mepivacaine, Prilocaine, Etidocaine. Miscellaneous : Phenacaine, Diperodon, Dibucaine.* Please follow the link  Local Anesthetics  

4.6 Thyroid and antithyroid drugs L-Thyroxine, L-Thyronine, Propylthiouracil, Methimazole. Please follow the link Presentation:  Thyroid Hormones                                    Youtube Video:  Thyroid Animation                                     Youtube Video:  Thyroid Hormone Synthesis and Antithyroid drugs

  4.2 Sex hormones : Testosterone, Nandralone, Progestrones, Oestriol, Oestradiol,Oestrione, Diethyl stilbestrol. Please follow the link   Sex hormones 4.3 Drugs for erectile dysfunction: Sildenafil, Tadalafil Please follow the link  Drugs for erectile dysfunction 4.4 Oral contraceptives: Mifepristone, Norgestril, Levonorgestrol Please follow the link  Oral contraceptives

 4.5 Corticosteroids Cortisone, Hydrocortisone, Prednisolone, Betamethasone,Dexamethasone Please follow the link  Adrenocorticoids or Corticoids

4.1 Drugs acting on Endocrine system Nomenclature, Stereochemistry and metabolism of steroids Please follow the links Steroid Nomenclature and stereochemistry Wilson and Gisvold’s Textbook Introduction of steroids  Steroid Assignment follow the link to complete the assignment Steroid Assignment-5   with answer supplement